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Harnessing RIBOnucleic acid - Small molecules Structures

Illustration - complex

Complex 2l94

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Pocket colors by molecule type

 RNA

 Protein

 DNA

These colors appear when a pocket is selected (the structure fades to show the pocket surface). Colors from the molecule-type palette (RNA / protein / DNA).

System information

Experimental technique Solution NMR
Experimental resolution N/A
System mass 14.86 kDa
Deposition year 2011
Molecule type RNA
# RNA entities 1
Organism Lentivirus
RCSB PDB Entry 2l94
Reference Marcheschi Ryan J., Tonelli Marco, Kumar Arvind, Butcher Samuel E.. 2011. Structure of the HIV-1 Frameshift Site RNA Bound to a Small Molecule Inhibitor of Viral Replication ACS Chemical Biology
Molecular Dynamics Simulation mmb-A01WQ, mmb-A01X1, mmb-A01XH, mmb-A022K, mmb-A022Q
Equivalence Class NR_all_80173.1
BGSU version: 4.52

Pockets List

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Cell colors for SiteScore and D Score:

 Favourable

 Intermediate

 Unfavourable

 Not available

ScoreThresholdMeaning
SiteScore< 0.8Non-drug binding site
SiteScore0.8 – 1.0Potential drug binding site
SiteScore> 1.0Promising binding site
D Score< 0.83Undruggable
D Score0.83 – 0.98Difficult
D Score> 0.98Druggable

Tick a pocket below to highlight it in the 3D structure above.

Compound L94
Residue . / 46
Chain B / A
Non-redundant True
Interacting RNA chains A/A
RNA environment detailled RNA-only
RNA environment global RNA
RNA family chains A/A: TAR_rna
RNA family global TAR_rna
Volume 164.64 Å3
Hydrophobicity 0.026
Hydrophilicity 0.867
Buriedness 0.653
Don/acc character 2.346
SiteScore 0.780
D Score 0.570
Kd 360uM