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Harnessing RIBOnucleic acid - Small molecules Structures

Illustration - complex

Complex 8eos

Legend

Pocket colors by molecule type

 RNA

 Protein

 DNA

These colors appear when a pocket is selected (the structure fades to show the pocket surface). Colors from the molecule-type palette (RNA / protein / DNA).

System information

Experimental technique Electron Microscopy
Experimental resolution 3.10
System mass 421.51 kDa
Deposition year 2022
Molecule type RNA/DNA/Protein
# RNA entities 1
Organism N/A
RCSB PDB Entry 8eos
Reference Vishwakarma Rishi K., Qayyum M. Zuhaib, Babitzke Paul, Murakami Katsuhiko S.. 2023. Allosteric mechanism of transcription inhibition by NusG-dependent pausing of RNA polymerase Proceedings of the National Academy of Sciences

Pockets List

Legend

Cell colors for SiteScore and D Score:

 Favourable

 Intermediate

 Unfavourable

 Not available

ScoreThresholdMeaning
SiteScore< 0.8Non-drug binding site
SiteScore0.8 – 1.0Potential drug binding site
SiteScore> 1.0Promising binding site
D Score< 0.83Undruggable
D Score0.83 – 0.98Difficult
D Score> 0.98Druggable

Tick a pocket below to highlight it in the 3D structure above.

Compound 2TM
Residue . / 1201
Chain J / C
Non-redundant True
Interacting RNA chains I/R
RNA environment detailled DNA, protein, ion
RNA environment global RNA/DNA/Protein
RNA family chains I/R: synthetic construct
RNA family global synthetic construct
Volume 347.46 Å3
Hydrophobicity 0.281
Hydrophilicity 1.279
Buriedness 0.845
Don/acc character 0.611
SiteScore 0.823
D Score 0.677
Kd